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39 Applicant: Quantum Genomics. Inventors : F. Balavoine, J-M Schneider, N.Couvrat, G. Coquerel, New crystalline phase of (3S,3S’) 4,4’-disulfanediylbis(3-aminobutane 1-sulfonic acid) with L-lysine. Filed the 22th of octobre 2012. EP 12306307.5.

38 Applicant: UNIVERSITY OF ROUEN. Inventors : Coquerel G., Sanselme M., Lafontaine A. Procédé de mesure de diffraction des rayons X, ses applications et dispositif de mise en oeuvre. International patent application PCT/FR2012/050707 (not yet published) filed on 02/04/2012 under priority filed on 6/04/2011.

37 Applicant: VIRO PHARMA. Inventors (and deposants for the US): Coquerel G., Levilain G., Petit M-N, Coste-Leconte S. Crystalline Phases of 5,6-Dichloro-2-(Isopropylamino)-(1-b-L-Ribofuranosyl)-1H-Benzimidazole. US Patent Application US20120178709 filed on 27/10/2011 under US Provisional application priority n° 61/407,622 filed on 28/10/2010

36 Applicant: QUANTUM GENOMICS. Inventors: Balavoine, F.; Madec, J.; Schneider, J.-M.; Coquerel, G.; Couvrat, N.; Cartigny, Y.; Petit, M.-N. Method for the preparation of (3S, 3S') 4, 4'-disulfanediylbis(3-aminobutane 1-sulfonic acid). International patent application WO2012/045849 filed on 07/10/2011 under priority filed on 07/10/2010.

35 Applicant: PCAS. Inventors: Chouippe S., Schneider J-M., Tauvel G., Coquerel G. Precursor phase and use thereof for preparing the magnesium salt tetrahydrate of an omeprazole enantiomer. European patent application EP2385046 filed on 29/04/2010 under priority filed on 03/05/2010.

34 Applicant: IPSEN PHARMA; Inventors: Mondoly, N.; Poirot, B.; Brochard, A.; Richard, J.; Delahaye, D.; Diolez, C.; Rolland, A.; Diancourt, F.; Coquerel, G.; Martins, D.; Linol, J.; Houssin, O.; Petit, M.-N.; Potter, B. V. L.; Woo, L. W. L. Compositions pharmaceutiques du 6-oxo-6,7,8,9,10,11-hexahydrocyclohepta 3-yl sulfamate; International patent application WO2010/092260 filed on 12/02/2010 under priority filed on 13/02/2009.

33 Applicant: POXEL; Inventors: Helmreich, M.; Niesert, C.-P.; Cravo, D.; Coquerel, G.; Levilain, G.; Wacharine-Antar, s.; Cardinaël, P. Process for enantiomeric separation of racemic dihydro-1, 3, 5 triazines via preferential crystallization. International patent application: WO2010/109015 filed on 26/03/2010 under priority filed on 26/03/2009.

32 Applicant: INNATE PHARMA. Inventors: Descamps, G.; Amharar, Y.; Cartigny, Y.; Coquerel, G. Novel Polymorphic form of CHDMAPP, method of preparation thereof, and pharmaceutical composition comprising same. International patent application WO2010/029062 filed on 08/09/2009 under priority filed on 10/09/2008.

31 Applicant: IPSEN PHARMA. Inventors: Delahaye, D.; Diolez, C.; Rolland, A.; Diancourt, F.; Brochard, A.; Mondoly, N.; Poirot, B.; Coquerel, G.; Martins, D.; Houssin, O.; Petit, M.-N. New polymorphic form, crystalline dimethyl sulfoxide solvate and crystalline 1, 4-dioxane hemisolvate of 6-oxo-6, 7, 8, 9, 10, 11-hexahydrocyclohepta(c)chromen-3-yl sulfamate, are steroid sulfatase inhibitors, useful to treat cancer. French patent application FR2942226 filed on 13/02/2009.

30 Applicant: IPSEN PHARMA. Inventors: Delahaye, D.; Diolez, C.; Rolland, A.; Diancourt, F.; Brochard, A.; Mondoly, N.; Poirot, B.; Coquerel, G.; Martins, D.; Linol, J.; Potter, B. V. L.; Woo, L. W. L. New polymorph of 6-oxo-6, 7, 8, 9, 10, 11-hexahydrocyclohepta(c) chromen-3-yl sulfamate having specific particle size, is steroid sulfatase inhibitor, useful to treat cancer and hormone-dependent cancers e.g. breast cancer. French patent application FR2942225 filed on 13/02/2009.

29 Applicant: SERVIER; Inventors: Martins, D.; Coquerel, G.; Linol, J.; Langlois, P. Novel process for obtaining the crystalline form V of Agomelatine. International patent application WO2010/015747 filed on 04/08/2009 under priority filed on 05/08/2008.

28 Applicant: UNIVERSITY OF ROUEN. Inventors: Levilain, G.; Coquerel, G. Process for the resolution of enantiomers by preferential evaporative crystallization. International patent application WO2011/07330 filed on 16/12/2010 under priorities filed on 18/12/2009 and 21/12/2009.

27 Applicant: UNIVERSITY OF ROUEN. Inventors : Coquerel, G.; Tauvel, G.; Petit, M.-N. Method for splitting omeprazole salts. International patent application WO 2009/027614 filed on 29/08/2008 under priority filed on 29/08/2007.

26 Applicant: SERVIER. Inventors: Coquerel, G.; Linol, J.; Le Pape, L.; Lecouvé, J.-P. Novel crystalline form VI of agomelatine, method for preparing same and pharmaceutical compositions containing same. International patent application WO2009/095555 filed on 07/11/2008 under priority filed on 09/11/2007.

25 Applicant: SANOFI AVENTIS. Inventors: Coquerel, G.; Fours, B. Isopropanol solvate of rimonabant, preparation method thereof and pharmaceutical compositions containing same. International patent application WO2009/050354 filed on 04/08/2008 under priority filed on 06/08/2007.

24 Applicant: SANOFI AVENTIS. Inventors: Coquerel, G.; Fours, B. 3-methylbutan-1-ol solvate of rimonabant, preparation method thereof and pharmaceutical compositions containing same. International patent application WO2009/050353 filed on 04/08/2008 under priority filed on 06/08/2007.

23 Applicant: SANOFI AVENTIS. Inventors: Coquerel, G.; Fours, B. Rimonabant 1, 4-dioxane solvate, method for preparing same and pharmaceutical compositions containing same. International patent application WO2009/053548 filed on 04/08/2008 under priority filed on 06/08/2007.

22 Applicant: SANOFI AVENTIS. Inventors: Coquerel, G.; Fours, B. Rimonabant 2-methoxyethanol solvate and method for preparing same. International patent application WO2009/053553 filed on 04/08/2008 under priority filed on 06/08/2007.

21 Applicant: SANOFI AVENTIS. Inventors: Coquerel, G.; Fours, B. Rimonabant DMSO solvate, method for preparing same and pharmaceutical compositions containing same. International patent application WO2009/053549 filed on 04/08/2008 under priority filed on 06/08/2007.

20 Applicant: SANOFI AVENTIS. Inventors: Coquerel, G.; Fours, B. Rimonabant N, N-dimethylformamide solvate, and method for preparing same. International patent application WO2009/053551 filed on 04/08/2008 under priority filed on 06/08/2007.

19 Applicant: SANOFI AVENTIS. Inventors: Coquerel, G.; Fours, B. Rimonabant N-methylpyrrolidone solvate, method for preparing same and pharmaceutical compositions containing same. International patent application WO2009/053550 filed on 04/08/2008 under priority filed on 06/08/2007.

18 Applicant: SANOFI AVENTIS. Inventors: Coquerel, G.; Duplaa, H.; Fours, B.; Monnier, O.; Ochsenbein, P. Rimonabant monohydrate, process for the preparation thereof and pharmaceutical compositions containing same. International patent application WO2007/090949 filed on 04/02/2007 under priority filed on 08/02/2006.

17 Applicant: SIDEM PHARMA. Inventors: Cohen, A.; Schutze, F.; Charbit, S.; Bernad, S.; Tauvel, G.; Petit, M.-N.; Coquerel, G. Conglomerates of tenatoprazole potassium salts. International patent application WO2008/081104 filed on 03/12/2007 under priority filed on 04/12/2006.

16 Applicant: SERVIER. Inventors: Coquerel, G.; Lefèbvre, L.; Souvie, J.-C.; Authouart, P. a crystalline form of the arginine salt of perindopril, process for preparing it, and pharmaceutical compositions comprising it. International patent application WO2007/099217 filed on 26/02/2007 under priority filed on 28/02/2006.

15 Applicant: SERVIER. Inventors: Coquerel, G.; Lefèbvre, L.; Souvie, J.-C.; Authouart, P. ss-crystalline form of perindopril arginine salt, method for making same, and pharmaceutical compositions containing same. International patent application WO2007/099216 filed on 26/02/2007 under priority filed on 28/02/2006.

14 Applicant: SERVIER. Inventors: Coquerel, G. ; Linol, J. ; Souvie J-C. nouvelle forme cristalline III de l'agomélatine, son procédé de préparation et les compositions pharmaceutiques qui la contiennent. International patent application WO2007/015003 filed on 02/08/2006 under priority filed on 03/08/2005.

13 Applicant: SERVIER. Inventors: Coquerel, G. ; Linol, J. ; Souvie J-C. Nouvelle forme cristalline IV de l'agomélatine, son procédé de préparation et les compositions pharmaceutiques qui la contiennent. International patent application WO2007/015002 filed on 02/08/2006 under priority filed on 03/08/2005.

12 Applicant: SERVIER. Inventors: Coquerel, G. ; Linol, J. ; Souvie J-C. Nouvelle forme cristalline V de l'agomélatine, son procédé de préparation et les compositions pharmaceutiques qui la contiennent. International patent application WO2007/015004 filed on 02/08/2006 under priority filed on 03/08/2005.

11 Applicant: INNATE PHARMA. Inventors: Coquerel, G.; Aubin, E. Phosphoantigen Salts of Organic Bases and Methods for their Crystallization. Purification by means of crystallization of some Pyrophosphate analogous antigen. International patent application WO2007/039635 filed on 05/10/2006 under priority filed on 06/10/2005.

10 Applicant: BIOPROJET. Inventors (and deposants for the US): Capet, M.; Coquerel, G.; Danvy, D.; Lecomte, J.-M.; Petit, M.-N.; Schwartz, J. C. Polymorphic forms of Fasidotril, their methods of preparation and pharmatical compositions comprising them. US Patent application US 6,767,921 filed on 26/03/2003 under priority filed on 29/03/2002.

09 Applicant: CEPHALON. Inventors : Broquaire, M.; Courvoisier, L.; Mallet, F.; Coquerel, G.; Frydman, A. Modafinil Polymorphic forms. International Patent application WO2004/014846 filed on 08/08/2003 under priorities filed on 09/08/2002 and 07/08/2003.

08 Applicant: CEPHALON. Inventors : Neckebrock, O.; Courvoisier, L.; Graf, S.; Serrure, G.; Coquerel, G.; Rose, S.; Besselièvre, C. Method for preparation of modafinil enantiomers and crystalline forms of optical enantiomers of modafinil. International Patent application 0

07 Applicant: CEPHALON. Inventors(and deposants for the US): Broquaire, M.; Courvoisier, L.; Branger-Zagouri, C.; Rose, S.; Coquerel, G. Polymorphic forms and solvates of -Modafinil. US provisional patent application n°60/402064 filed on 08/09/ 2002.

06 Applicant: SERVIER. Inventors : Pfeiffer, B.; Ginot, Y.-M.; Coquerel, G.; Beilles, S. Nouvelle forme cristalline "alpha" du sel de ter-butylamine du perindopril, son procédé de fabrication, et les compositions pharmaceutiques qui la contiennent. International Patent Application WO2001/087835 filed on 06/07/2001 under priority filed on 06/07/2000.

05 Applicant: SERVIER. Inventors : Pfeiffer, B.; Ginot, Y.-M.; Coquerel, G.; Beilles, S. Nouvelle forme "béta" du del de ter-butylamine du perindopril, son procédé de préparation, et les compositions pharmaceutiques qui la contiennent. International Patent Application WO2001/087836 filed on 06/07/2001 under priority filed on 06/07/2000.

04 Applicant: SERVIER. Inventors : Pfeiffer, B.; Ginot, Y.-M.; Coquerel, G.; Beilles, S. Nouvelle forme cristalline "gamma" de sel de ter-butylamine du perindopril, son procédé de préparation, et les compositions pharmaceutiques qui la contiennent. International Patent Application WO2001/087839 filed on 06/07/2001 under priority filed on 06/07/2000.

03 Applicant: UNIVERSITY OF ROUEN. Inventors: Coquerel, G.; Catroux, L.; Combret, Y. Procédé de dédoublement par diastéréoisomères et par cristallisation préférentielle dans la série des 1-amino-alcan-2-ols. International Patent application WO1998/023559 filed on 28/11/1997 under priority filed on 28/11/1996.

02 Applicant: UNIVERSITY OF ROUEN. Inventors: Coquerel, G.; Petit, M.-N.; Bouaziz, R. Procédé de dédoublement (AS3PC) de deux antipodes optiques par entraînement polythermique programmé et auto-ensemencé. International Patent application WO1995/008522 filed on 22/09/1994 under priority filed on 23/09/1993.

01 Applicant: JOUVEINAL. Inventors: Depernet, D.; Bouaziz, R.; Coquerel, G.; Petit, M.-N. Procédé de dédoublement d'hydantoïnes chirales. WO1992/008702 filed on 15/11/1991 under priority filed on 16/11/1990.